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- W2510029653 abstract "Abstract Trace amine-associated receptors (TAARs) are a vertebrate, G-protein-coupled, family of receptors found throughout the body. Within the CNS, TAAR1, for which the endogenous trace amines p-tyramine and 2-phenylethylamine are high-affinity agonists, activation has been shown to decrease dopaminergic tone, an effect mediated via regulation of both pre- and postsynaptic D2-like dopamine receptors. This occurs in a biased manner, with only the β-arrestin signaling pathway modified. Consistent with this, TAAR1 agonists decrease the self-administration and reinforcing properties of various drugs of abuse, and exhibit an activity profile predictive of beneficial effects in schizophrenia. There is also evidence that TAAR1 may play a role in controlling energy metabolism, although whether this is mediated centrally or peripherally is unknown. All TAAR, with the exception of TAAR1, also function as olfactory receptors mediating innate behavioral responses to various conspecific and heterospecific urinary cues." @default.
- W2510029653 created "2016-09-16" @default.
- W2510029653 creator A5015490085 @default.
- W2510029653 date "2016-01-01" @default.
- W2510029653 modified "2023-09-25" @default.
- W2510029653 title "Trace Amines and Their Receptors in the Control of Cellular Homeostasis" @default.
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