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- W2524374821 abstract "Publisher Summary This chapter demonstrates that molecular biology of GABAA receptors in the central nervous system (CNS) has demonstrated remarkable heterogeneity in the expression of unique GABA isoreceptors. Detailed studies on the distribution of GABAA receptor subunits throughout the brain elucidate the subunit composition of isoreceptors present in various cell populations. Studies on the effects of various neuropharmacological agents on the expression of these subunits may elucidate how each of the subunits is regulated and how alterations in the expression of various subunits affect the function of various GABAA isoreceptors. The complexity of GABAA isoreceptors in the mammalian CNS explains the diverse effects of chronic benzodiazepine, barbiturate, and ethanol administration on GABAA receptor binding sites. Identification of the actual binding sites for GABAA/benzodiazepine ligands will help identify the GABAA isoreceptors/ subunits that are labeled by each of the available radioligands. Anxiety, epilepsy, depression, and other mood disorders may be ameliorated by interventions in the structure, function, and regulation of GABAA receptors." @default.
- W2524374821 created "2016-10-07" @default.
- W2524374821 creator A5024081434 @default.
- W2524374821 date "1995-01-01" @default.
- W2524374821 modified "2023-09-26" @default.
- W2524374821 title "Regulation of GABAA Receptor Function and Gene Expression in the Central Nervous System" @default.
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