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- W2531384287 abstract "Aim: In this study, we constructed a novel vector (BioPf-M-loaded Alg-microparticles [Alg-BioPf-M]) with nano-in-micro structure to improve the oral absorption of docetaxel (DTX) by sequentially dual-targeting functions toward intestine and sodium-dependent multivitamin transporter based on entrapping biotin-modified micelles into alginate microparticles. Methods: A series of characteristics of this system was investigated, such as drug release, cellular uptake, transport pathway and the comprehensive in vivo studies including pharmacokinetic studies, anti-tumor activity and toxicity study. Results: The bioavailability of DTX-loaded Alg-BioPf-M was 27.4-fold higher than that of free DTX after oral administration and achieved superior tumor inhibition of 84.6% against sarcoma 180 tumors. Conclusion: These results demonstrated that the Alg-BioPf-M was a promising vector for oral delivery of DTX." @default.
- W2531384287 created "2016-10-21" @default.
- W2531384287 creator A5002288726 @default.
- W2531384287 creator A5025799914 @default.
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- W2531384287 date "2016-12-01" @default.
- W2531384287 modified "2023-10-13" @default.
- W2531384287 title "Sequentially dual-targeting vector with nano-in-micro structure for improved docetaxel oral delivery <i>in vivo</i>" @default.
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- W2531384287 doi "https://doi.org/10.2217/nnm-2016-0259" @default.
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