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- W2566029877 abstract "Peroxisome proliferator-activated receptor α (PPARα) plays a key role in lipid metabolism and glucose homeostasis and a crucial role in the prevention and treatment of metabolic diseases. Natural dietary compounds, including nutrients and phytochemicals, are PPARα ligands or modulators. High-throughput screening assays have been developed to screen for PPARα ligands and modulators in our diet. In the present review, we discuss recent advances in our knowledge of PPARα, including its structure, function, and ligand and modulator screening assays, and summarize the different types of dietary PPARα ligands and modulators. 过氧化物酶体增殖物活化受体α(PPARα)在调节脂质代谢和维持糖代谢稳态过程中起到重要作用,同时在预防及治疗代谢性疾病中发挥着关键作用。很多天然食物源化合物,包括营养素及植物化学物,都是PPARα的配体或调节剂。对于食源性PPARα配体或调节剂目前已有多种高通量筛选方法。本文讨论了PPARα的结构、功能及其配体或调节剂的筛选方法,同时还总结了目前发现的来自食物中不同种类的PPARα配体和调节剂。" @default.
- W2566029877 created "2017-01-06" @default.
- W2566029877 creator A5023085226 @default.
- W2566029877 creator A5060969271 @default.
- W2566029877 creator A5091188597 @default.
- W2566029877 date "2016-12-22" @default.
- W2566029877 modified "2023-10-18" @default.
- W2566029877 title "Peroxisome proliferator-activated receptor<b>α</b>ligands and modulators from dietary compounds: Types, screening methods and functions" @default.
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- W2566029877 doi "https://doi.org/10.1111/1753-0407.12506" @default.
- W2566029877 hasPubMedId "https://pubmed.ncbi.nlm.nih.gov/27863018" @default.
- W2566029877 hasPublicationYear "2016" @default.
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