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- W2600487630 abstract "Type 2 diabetes mellitus is a progressive disease with multiple underlying pathophysiologic defects. Monotherapy alone cannot maintain glycemic control and leads to treatment failure. Ideally, a combination of glucose-lowering agents should have complementary mechanisms of action that address multiple pathophysiologic pathways, can be used at all stages of the disease, and be generally well tolerated with no increased risk of hypoglycemia, cardiovascular events, or weight gain. The combination should also provide conveniences for patients, such as oral dosing, single-pill formulations, and once-daily administration, potentially translating to improved adherence. Two classes of glucose-lowering agents that meet these criteria are the sodium glucose cotransporter-2 (SGLT2) inhibitors and dipeptidyl peptidase-4 (DPP-4) inhibitors. This article reviews the rationale for combination therapy with these agents, and evidence from clinical trials with empagliflozin and linagliptin or dapagliflozin and saxagliptin in the management of type 2 diabetes mellitus. Both combinations have been approved as single-pill formulations." @default.
- W2600487630 created "2017-04-07" @default.
- W2600487630 creator A5084556839 @default.
- W2600487630 date "2017-04-03" @default.
- W2600487630 modified "2023-09-25" @default.
- W2600487630 title "SGLT2 inhibitor/DPP-4 inhibitor combination therapy – complementary mechanisms of action for management of type 2 diabetes mellitus" @default.
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- W2600487630 doi "https://doi.org/10.1080/00325481.2017.1307081" @default.
- W2600487630 hasPubMedId "https://pubmed.ncbi.nlm.nih.gov/28322073" @default.
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