Matches in SemOpenAlex for { <https://semopenalex.org/work/W2605669685> ?p ?o ?g. }
Showing items 1 to 96 of
96
with 100 items per page.
- W2605669685 endingPage "2342" @default.
- W2605669685 startingPage "2338" @default.
- W2605669685 abstract "The P2X3 receptor is primarily expressed in the peripheral sensory nerves, and therefore, antagonists of this receptor may be useful for the treatment of chronic pain. Pyrrolinone derivatives have been identified as a novel class of P2X3 receptor antagonists. A lead structure with moderate activity was discovered through a high-throughput screening assay. A structure-activity study led to the discovery of several P2X3 receptor antagonists. Compound 34 showed potent and specific antagonistic activity and analgesic efficacy." @default.
- W2605669685 created "2017-04-28" @default.
- W2605669685 creator A5000190193 @default.
- W2605669685 creator A5002445981 @default.
- W2605669685 creator A5009929660 @default.
- W2605669685 creator A5013156919 @default.
- W2605669685 creator A5016747876 @default.
- W2605669685 creator A5034040324 @default.
- W2605669685 creator A5040030946 @default.
- W2605669685 creator A5050088505 @default.
- W2605669685 creator A5063380148 @default.
- W2605669685 creator A5076959343 @default.
- W2605669685 creator A5077042490 @default.
- W2605669685 creator A5077307889 @default.
- W2605669685 creator A5079183925 @default.
- W2605669685 creator A5081995756 @default.
- W2605669685 date "2018-07-01" @default.
- W2605669685 modified "2023-09-27" @default.
- W2605669685 title "Pyrrolinone derivatives as a new class of P2X3 receptor antagonists. Part 1: Initial structure-activity relationship studies of a hit from a high throughput screening" @default.
- W2605669685 cites W1623121663 @default.
- W2605669685 cites W1975947882 @default.
- W2605669685 cites W2048201868 @default.
- W2605669685 cites W2063781307 @default.
- W2605669685 cites W2084701217 @default.
- W2605669685 cites W2100452437 @default.
- W2605669685 cites W2106753138 @default.
- W2605669685 cites W2127376430 @default.
- W2605669685 cites W2156346381 @default.
- W2605669685 cites W2470301777 @default.
- W2605669685 cites W2950813711 @default.
- W2605669685 doi "https://doi.org/10.1016/j.bmcl.2017.04.060" @default.
- W2605669685 hasPubMedId "https://pubmed.ncbi.nlm.nih.gov/29805055" @default.
- W2605669685 hasPublicationYear "2018" @default.
- W2605669685 type Work @default.
- W2605669685 sameAs 2605669685 @default.
- W2605669685 citedByCount "7" @default.
- W2605669685 countsByYear W26056696852019 @default.
- W2605669685 countsByYear W26056696852020 @default.
- W2605669685 countsByYear W26056696852021 @default.
- W2605669685 crossrefType "journal-article" @default.
- W2605669685 hasAuthorship W2605669685A5000190193 @default.
- W2605669685 hasAuthorship W2605669685A5002445981 @default.
- W2605669685 hasAuthorship W2605669685A5009929660 @default.
- W2605669685 hasAuthorship W2605669685A5013156919 @default.
- W2605669685 hasAuthorship W2605669685A5016747876 @default.
- W2605669685 hasAuthorship W2605669685A5034040324 @default.
- W2605669685 hasAuthorship W2605669685A5040030946 @default.
- W2605669685 hasAuthorship W2605669685A5050088505 @default.
- W2605669685 hasAuthorship W2605669685A5063380148 @default.
- W2605669685 hasAuthorship W2605669685A5076959343 @default.
- W2605669685 hasAuthorship W2605669685A5077042490 @default.
- W2605669685 hasAuthorship W2605669685A5077307889 @default.
- W2605669685 hasAuthorship W2605669685A5079183925 @default.
- W2605669685 hasAuthorship W2605669685A5081995756 @default.
- W2605669685 hasConcept C170493617 @default.
- W2605669685 hasConcept C185592680 @default.
- W2605669685 hasConcept C193042331 @default.
- W2605669685 hasConcept C202751555 @default.
- W2605669685 hasConcept C2776885963 @default.
- W2605669685 hasConcept C2780820201 @default.
- W2605669685 hasConcept C51323132 @default.
- W2605669685 hasConcept C55493867 @default.
- W2605669685 hasConcept C71924100 @default.
- W2605669685 hasConcept C98274493 @default.
- W2605669685 hasConceptScore W2605669685C170493617 @default.
- W2605669685 hasConceptScore W2605669685C185592680 @default.
- W2605669685 hasConceptScore W2605669685C193042331 @default.
- W2605669685 hasConceptScore W2605669685C202751555 @default.
- W2605669685 hasConceptScore W2605669685C2776885963 @default.
- W2605669685 hasConceptScore W2605669685C2780820201 @default.
- W2605669685 hasConceptScore W2605669685C51323132 @default.
- W2605669685 hasConceptScore W2605669685C55493867 @default.
- W2605669685 hasConceptScore W2605669685C71924100 @default.
- W2605669685 hasConceptScore W2605669685C98274493 @default.
- W2605669685 hasIssue "13" @default.
- W2605669685 hasLocation W26056696851 @default.
- W2605669685 hasLocation W26056696852 @default.
- W2605669685 hasOpenAccess W2605669685 @default.
- W2605669685 hasPrimaryLocation W26056696851 @default.
- W2605669685 hasRelatedWork W2002661198 @default.
- W2605669685 hasRelatedWork W2012391196 @default.
- W2605669685 hasRelatedWork W2018762970 @default.
- W2605669685 hasRelatedWork W2020881343 @default.
- W2605669685 hasRelatedWork W2043685761 @default.
- W2605669685 hasRelatedWork W2051684012 @default.
- W2605669685 hasRelatedWork W2147753672 @default.
- W2605669685 hasRelatedWork W2272504806 @default.
- W2605669685 hasRelatedWork W4318830844 @default.
- W2605669685 hasRelatedWork W2188272290 @default.
- W2605669685 hasVolume "28" @default.
- W2605669685 isParatext "false" @default.
- W2605669685 isRetracted "false" @default.
- W2605669685 magId "2605669685" @default.
- W2605669685 workType "article" @default.