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- W2607029183 endingPage "104" @default.
- W2607029183 startingPage "91" @default.
- W2607029183 abstract "Thyroid hormones (THs) play key roles in modulating the overall metabolism of the body, protein synthesis, fat metabolism, neuronal and bone growth, and cardiovascular as well as renal functions. In this review, we discuss on the thyroid hormone synthesis and activation, thyroid hormone receptors (TRs) and mechanism of action, applications of thyroid hormone analogues, particularly the compounds that are selective ligands for TRβ receptors, or enzyme inhibitors for the treatment of thyroidal disorders with a specific focus on thyroid peroxidase and iodothyronine deiodinases. We also discuss on the development of small-molecule deiodinase mimetics and their mechanism of deiodination, as these compounds have the potential to regulate the thyroid hormone levels." @default.
- W2607029183 created "2017-04-28" @default.
- W2607029183 creator A5032638949 @default.
- W2607029183 creator A5068518494 @default.
- W2607029183 date "2017-12-01" @default.
- W2607029183 modified "2023-10-02" @default.
- W2607029183 title "Novel thyroid hormone analogues, enzyme inhibitors and mimetics, and their action" @default.
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