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- W2617260055 abstract "Medullary thyroid cancer accounts for less than 10% of all thyroid cancers.Aggressive metastatic forms of this disease however, are incurable and can cause significantsymptoms including diarrhea and pain. Hereditary and some sporadic forms of the diseaseare characterized by a mutation of the proto-oncogene RET. This results in an abnormal growthfactor receptor that, in turn, allows the malignant cells to survive and metastasize. New tyrosinekinase inhibitors have been shown to effectively target RET in vitro. One of the first of theseagents, vandetanib, has been evaluated in international Phase II and III clinical trials. In 2011,vandetanib became the first agent approved by the US FDA for use in metastatic medullarythyroid cancer. This article examines the clinical use of this agent" @default.
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- W2617260055 date "2013-01-01" @default.
- W2617260055 modified "2023-09-23" @default.
- W2617260055 title "Vandetanib for aggressive andsymptomatic medullary thyroid cancer" @default.
- W2617260055 hasPublicationYear "2013" @default.
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