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- W2621670189 abstract "The PPARs are a subfamily of three ligand-inducible transcription factors, which belong to the superfamily of nuclear hormone receptors. In mammals, the PPAR subfamily consists of three members: PPAR-α, PPAR-β/δ and PPAR-γ. PPARs control the expression of a large number of genes involved in metabolic homeostasis, lipid, glucose and energy metabolism, adipogenesis and inflammation. PPARs regulate a large number of metabolic pathways that are implicated in the pathogenesis of metabolic diseases such as metabolic syndrome, Type 2 diabetes mellitus, nonalcoholic fatty liver disease and cardiovascular disease. The aim of this review is to provide up-to-date information about the biochemical and metabolic actions of PPAR-β/δ and PPAR-γ, the therapeutic potential of their agonists currently under clinical development and the cardiovascular disease outcome of clinical trials of PPAR-γ agonists, pioglitazone and rosiglitazone." @default.
- W2621670189 created "2017-06-15" @default.
- W2621670189 creator A5050996840 @default.
- W2621670189 creator A5053011805 @default.
- W2621670189 creator A5059308494 @default.
- W2621670189 creator A5077425218 @default.
- W2621670189 creator A5079453429 @default.
- W2621670189 date "2017-05-01" @default.
- W2621670189 modified "2023-10-09" @default.
- W2621670189 title "PPARs: regulators of metabolism and as therapeutic targets in cardiovascular disease. Part II: PPAR-β/δ and PPAR-γ" @default.
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