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- W2743170615 abstract "Galeterone is a steroid 17-α-hydroxylase/17,20 lyase and androgen receptor antagonist intended for patients with prostate cancer. Similar to abiraterone, galeterone has a steroid scaffold structure and mimics natural ligands; thus, these agents are metabolized by the same enzymes that synthesize or degrade naturally occurring steroids, which can result in attenuated efficacy." @default.
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- W2743170615 date "2017-08-08" @default.
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- W2743170615 title "The influence of steroid metabolism on CYP17A1 inhibitor activity" @default.
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- W2743170615 doi "https://doi.org/10.1038/nrurol.2017.132" @default.
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