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- W274997347 endingPage "190" @default.
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- W274997347 abstract "Abstract The liver X receptors (LXR) are crucial regulators of metabolism. After ligand binding, they regulate gene transcription and thereby mediate changes in metabolic pathways. Modulation of LXR and their downstream targets has appeared to be a promising treatment for metabolic diseases especially atherosclerosis and cholesterol metabolism. However, the complexity of LXR action in various metabolic tissues and the liver side effect of LXR activation have slowed down the interest for LXR drugs. In this review, we summarized the role of LXR in the main metabolically active tissues with a special focus on obesity and associated diseases in mammals. We will also discuss the dual interplay between the two LXR isoforms suggesting that they may collaborate to establish a fine and efficient system for the maintenance of metabolism homeostasis." @default.
- W274997347 created "2016-06-24" @default.
- W274997347 creator A5026937087 @default.
- W274997347 creator A5085801141 @default.
- W274997347 date "2015-05-06" @default.
- W274997347 modified "2023-10-09" @default.
- W274997347 title "Liver X receptors as regulators of metabolism" @default.
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