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- W2753766712 endingPage "604" @default.
- W2753766712 startingPage "585" @default.
- W2753766712 abstract "Epigenetic mechanisms, including DNA methylation and posttranslational histone modifications, play a pivotal role in DNA replication/repair and gene expression regulation. These epigenetic mechanisms are responsible for controlling cellular functions, such as cell cycle progression, immunoresponse, and signal transduction. Among the epigenetic mechanisms, the methylation of DNA and histones is closely associated with the oncogenesis and proliferation of cancer cells, and alterations of DNA methylation and histone methylation have been identified in many cancer cells. Several enzymes that control the methylation of DNA or histones have been identified, including DNA methyltransferases, ten-eleven translocation proteins, lysine methyltransferases, lysine demethylases, protein arginine methyltransferases, and peptidyl arginine deiminases. As some of the enzymes are involved in cancer, their inhibitors are considered useful not only as chemical tools for probing the biology of DNA and histone methylation, but also as anticancer agents. In this chapter, hitherto reported enzyme inhibitors are presented and their potential as anticancer agents is discussed." @default.
- W2753766712 created "2017-09-15" @default.
- W2753766712 creator A5044997693 @default.
- W2753766712 date "2017-01-01" @default.
- W2753766712 modified "2023-09-27" @default.
- W2753766712 title "DNA and Histone Modifications in Cancer Therapy" @default.
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