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- W2756935148 endingPage "12474" @default.
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- W2756935148 abstract "Natural products have served as powerful therapeutics against pathogenic bacteria since the golden age of antibiotics of the mid-20th century. However, the increasing frequency of antibiotic-resistant infections clearly demonstrates that new antibiotics are critical for modern medicine. Because combinatorial approaches have not yielded effective drugs, we propose that the development of new antibiotics around proven natural scaffolds is the best short-term solution to the rising crisis of antibiotic resistance. We analyze herein synthetic approaches aiming to reengineer natural products into potent antibiotics. Furthermore, we discuss approaches in modulating quorum sensing and biofilm formation as a nonlethal method, as well as narrow-spectrum pathogen-specific antibiotics, which are of interest given new insights into the implications of disrupting the microbiome." @default.
- W2756935148 created "2017-10-06" @default.
- W2756935148 creator A5023759374 @default.
- W2756935148 creator A5072469847 @default.
- W2756935148 creator A5073672011 @default.
- W2756935148 date "2017-09-27" @default.
- W2756935148 modified "2023-10-17" @default.
- W2756935148 title "Natural Products as Platforms To Overcome Antibiotic Resistance" @default.
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