Matches in SemOpenAlex for { <https://semopenalex.org/work/W2789808439> ?p ?o ?g. }
- W2789808439 abstract "Abstract Transcription factors regulate gene expression in cells and control cellular development, function, and death. Dysregulation of transcription factors is often associated with disease, including cancer. As such, transcription factors are attractive targets for design of therapeutics against disease. Transcription factors function using protein‐protein and protein‐DNA interactions that occur over relatively large surface areas: this lack of a small and defined “ligand binding site” has proven to be challenging to target with small molecules. Peptide therapeutics, therefore, provide an alternate approach toward design of inhibitory agents. Transcription factors are conveniently modular by design: just the small domain that is responsible for the transcription factor's DNA binding or a protein‐protein interaction or another function, can serve as the basis for novel peptide therapeutics. In this review, examples of peptides that directly interfere with transcription factors will be discussed." @default.
- W2789808439 created "2018-03-29" @default.
- W2789808439 creator A5044146971 @default.
- W2789808439 creator A5058640045 @default.
- W2789808439 date "2018-02-10" @default.
- W2789808439 modified "2023-10-16" @default.
- W2789808439 title "Peptide therapeutics that directly target transcription factors" @default.
- W2789808439 cites W1550069159 @default.
- W2789808439 cites W1574155225 @default.
- W2789808439 cites W1584683177 @default.
- W2789808439 cites W1597158509 @default.
- W2789808439 cites W1633256579 @default.
- W2789808439 cites W1940451643 @default.
- W2789808439 cites W1964369521 @default.
- W2789808439 cites W1965638470 @default.
- W2789808439 cites W1974521227 @default.
- W2789808439 cites W1988929415 @default.
- W2789808439 cites W1989162648 @default.
- W2789808439 cites W1989467084 @default.
- W2789808439 cites W1989557252 @default.
- W2789808439 cites W1990320777 @default.
- W2789808439 cites W1991647220 @default.
- W2789808439 cites W1991780615 @default.
- W2789808439 cites W1992450378 @default.
- W2789808439 cites W2004361605 @default.
- W2789808439 cites W2006833515 @default.
- W2789808439 cites W2006885289 @default.
- W2789808439 cites W2008223493 @default.
- W2789808439 cites W2010117150 @default.
- W2789808439 cites W2013016540 @default.
- W2789808439 cites W2014740187 @default.
- W2789808439 cites W2017580443 @default.
- W2789808439 cites W2021536610 @default.
- W2789808439 cites W2022320757 @default.
- W2789808439 cites W2023697479 @default.
- W2789808439 cites W2024689678 @default.
- W2789808439 cites W2028275307 @default.
- W2789808439 cites W2029012405 @default.
- W2789808439 cites W2029215616 @default.
- W2789808439 cites W2032023033 @default.
- W2789808439 cites W2035777673 @default.
- W2789808439 cites W2037438619 @default.
- W2789808439 cites W2037471080 @default.
- W2789808439 cites W2038720675 @default.
- W2789808439 cites W2042061022 @default.
- W2789808439 cites W2042143995 @default.
- W2789808439 cites W2044365745 @default.
- W2789808439 cites W2051409637 @default.
- W2789808439 cites W2054616775 @default.
- W2789808439 cites W2060846993 @default.
- W2789808439 cites W2061183445 @default.
- W2789808439 cites W2065292885 @default.
- W2789808439 cites W2066525432 @default.
- W2789808439 cites W2081314633 @default.
- W2789808439 cites W2082493554 @default.
- W2789808439 cites W2085609942 @default.
- W2789808439 cites W2090471601 @default.
- W2789808439 cites W2091770992 @default.
- W2789808439 cites W2093279074 @default.
- W2789808439 cites W2094784156 @default.
- W2789808439 cites W2095205674 @default.
- W2789808439 cites W2099132605 @default.
- W2789808439 cites W2101143531 @default.
- W2789808439 cites W2102154371 @default.
- W2789808439 cites W2111670964 @default.
- W2789808439 cites W2112916046 @default.
- W2789808439 cites W2113300574 @default.
- W2789808439 cites W2119483052 @default.
- W2789808439 cites W2122874647 @default.
- W2789808439 cites W2124690921 @default.
- W2789808439 cites W2126410372 @default.
- W2789808439 cites W2127321901 @default.
- W2789808439 cites W2127609327 @default.
- W2789808439 cites W2128888675 @default.
- W2789808439 cites W2133335149 @default.
- W2789808439 cites W2136007332 @default.
- W2789808439 cites W2140679819 @default.
- W2789808439 cites W2146556279 @default.
- W2789808439 cites W2147135207 @default.
- W2789808439 cites W2148515217 @default.
- W2789808439 cites W2151981602 @default.
- W2789808439 cites W2153598858 @default.
- W2789808439 cites W2155625886 @default.
- W2789808439 cites W2162723598 @default.
- W2789808439 cites W2165750540 @default.
- W2789808439 cites W2168717243 @default.
- W2789808439 cites W2171057750 @default.
- W2789808439 cites W2173231155 @default.
- W2789808439 cites W2183415805 @default.
- W2789808439 cites W2207542692 @default.
- W2789808439 cites W2273399293 @default.
- W2789808439 cites W2296805281 @default.
- W2789808439 cites W2341703160 @default.
- W2789808439 cites W2344125583 @default.
- W2789808439 cites W2404525374 @default.
- W2789808439 cites W2468743286 @default.
- W2789808439 cites W2493417617 @default.
- W2789808439 cites W2507443415 @default.
- W2789808439 cites W2522094723 @default.
- W2789808439 cites W2534930232 @default.