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- W2790773084 endingPage "554" @default.
- W2790773084 startingPage "534" @default.
- W2790773084 abstract "Glycopeptide antibiotics are drugs of last resort for treating severe infections caused by multi-drug resistant Gram-positive pathogens. First-generation glycopeptides (vancomycin and teicoplanin) are produced by soil-dwelling actinomycetes. Second-generation glycopeptides (dalbavancin, oritavancin, and telavancin) are semi-synthetic derivatives of the progenitor natural products. Herein, we cover past and present biotechnological approaches for searching for and producing old and new glycopeptide antibiotics. We review the strategies adopted to increase microbial production (from classical strain improvement to rational genetic engineering), and the recent progress in genome mining, chemoenzymatic derivatization, and combinatorial biosynthesis for expanding glycopeptide chemical diversity and tackling the never-ceasing evolution of antibiotic resistance." @default.
- W2790773084 created "2018-03-29" @default.
- W2790773084 creator A5015667865 @default.
- W2790773084 creator A5023715607 @default.
- W2790773084 creator A5081315059 @default.
- W2790773084 creator A5091255513 @default.
- W2790773084 date "2018-03-01" @default.
- W2790773084 modified "2023-10-07" @default.
- W2790773084 title "Old and new glycopeptide antibiotics: From product to gene and back in the post-genomic era" @default.
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