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- W2791792477 endingPage "581" @default.
- W2791792477 startingPage "581" @default.
- W2791792477 abstract "This review summarizes recent progress and developments as well as the most important pitfalls in targeted alpha-particle therapy, covering single alpha-particle emitters as well as in vivo alpha-particle generators. It discusses the production of radionuclides like 211At, 223Ra, 225Ac/213Bi, labelling and delivery employing various targeting vectors (small molecules, chelators for alpha-emitting nuclides and their biomolecular targets as well as nanocarriers), general radiopharmaceutical issues, preclinical studies, and clinical trials including the possibilities of therapy prognosis and follow-up imaging. Special attention is given to the nuclear recoil effect and its impacts on the possible use of alpha emitters for cancer treatment, proper dose estimation, and labelling chemistry. The most recent and important achievements in the development of alpha emitters carrying vectors for preclinical and clinical use are highlighted along with an outlook for future developments." @default.
- W2791792477 created "2018-03-29" @default.
- W2791792477 creator A5029805801 @default.
- W2791792477 creator A5038616265 @default.
- W2791792477 creator A5076490720 @default.
- W2791792477 date "2018-03-05" @default.
- W2791792477 modified "2023-10-14" @default.
- W2791792477 title "Progress in Targeted Alpha-Particle Therapy. What We Learned about Recoils Release from In Vivo Generators" @default.
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