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- W2793669837 endingPage "181" @default.
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- W2793669837 abstract "The Met proto-oncogene encodes MET tyrosine kinase protein which is a receptor for hepatocyte growth factor/scatter factor (HGF/SF). HGF binds to and activates MET to regulate diversified cellular and molecular activities such as proliferation, motility, differentiation, and survival. Aberration of HGF/MET signaling plays a proven role in promoting cancer initiation and malignant progression, providing a strong rationale for targeting the MET signaling pathway in the treatment of cancer. Several anti-HGF and anti-MET monoclonal antibodies, as well as small-molecule inhibitors of MET, are being evaluated in clinical trials for the treatment of various cancers. In this chapter, we discuss the role of HGF/MET signaling in cancer development and progression, the strategies for targeting MET signaling, as well as the promises and challenges of MET-targeted therapeutics." @default.
- W2793669837 created "2018-03-29" @default.
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- W2793669837 creator A5060311312 @default.
- W2793669837 creator A5067439838 @default.
- W2793669837 creator A5078666853 @default.
- W2793669837 date "2017-11-17" @default.
- W2793669837 modified "2023-10-15" @default.
- W2793669837 title "The HGF/MET Signaling and Therapeutics in Cancer" @default.
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