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- W2793720586 abstract "We prepared gadolinium oxide (Gd 2 O 3 ) nanoparticles (GNPs) coated with a trans‐activator of transcription (TAT) peptide with cell‐penetrating ability ( i.e ., TAT‐GNPs) through one‐pot process. We characterized the particle diameter, surface‐coating structure, water proton relaxivities, and in vitro cellular toxicities of the TAT‐GNPs. We measured in vivo T 1 magnetic resonance images (MRI) in a model nude mouse with liver cancer prior and posterior to intravenous administration. The average particle diameter of the GNPs was 1.5 nm. The sample solution exhibited a longitudinal water proton relaxivity (r 1 ) of 18.2/s/mM (r 2 /r 1 = 1.6, r 2 = transverse water proton relaxivity), which is four to five times higher than those of commercial Gd‐chelates. The in vivo T 1 MRI exhibited positively (or T 1 ) enhanced contrasts in the mouse liver cancer after intravenous administration, demonstrating that the TAT‐GNPs acted as an enhanced cancer‐imaging agent similar to the cancer‐targeting agent in T 1 MRI." @default.
- W2793720586 created "2018-03-29" @default.
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- W2793720586 date "2018-02-27" @default.
- W2793720586 modified "2023-09-23" @default.
- W2793720586 title "Synthesis, Characterization, and Enhanced Cancer-Imaging Application of Trans-activator of Transcription Peptide-conjugated Ultrasmall Gadolinium Oxide Nanoparticles" @default.
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- W2793720586 doi "https://doi.org/10.1002/bkcs.11404" @default.
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