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- W2793900979 endingPage "85" @default.
- W2793900979 startingPage "73" @default.
- W2793900979 abstract "DNA and histone methylation belong to the key regulatory components in the epigenetic machinery, and dysregulations of these processes have been associated with various human diseases. Small molecule modulators of these epigenetic targets are highly valuable both as chemical probes to study the biological roles of the target proteins, and as potential therapeutics. Indeed, recent years have seen the discovery of chemical modulators of several epigenetic targets, some of which are already marketed drugs or undergoing clinical trials. In this review, we will focus on small molecule modulators of DNA and histone methylation." @default.
- W2793900979 created "2018-03-29" @default.
- W2793900979 creator A5016266091 @default.
- W2793900979 creator A5019995093 @default.
- W2793900979 creator A5089212888 @default.
- W2793900979 date "2018-08-01" @default.
- W2793900979 modified "2023-10-14" @default.
- W2793900979 title "Epigenetic small molecule modulators of histone and DNA methylation" @default.
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