Matches in SemOpenAlex for { <https://semopenalex.org/work/W2801253218> ?p ?o ?g. }
- W2801253218 endingPage "152" @default.
- W2801253218 startingPage "147" @default.
- W2801253218 abstract "Drug-receptor interaction plays an important role in a series of biological effects, such as cell proliferation, immune response, tumor metastasis, and drug delivery. Therefore, the research on drug-receptor interaction is growing rapidly. The equilibrium dissociation constant (KD) is the basic parameter to evaluate the binding property of the drug-receptor. Thus, a variety of analytical methods have been established to determine the KD values, including radioligand binding assay, surface plasmon resonance method, fluorescence energy resonance transfer method, affinity chromatography, and isothermal titration calorimetry. With the invention and innovation of new technology and analysis method, there is a deep exploration and comprehension about drug-receptor interaction. This review discusses the different methods of determining the KD values, and analyzes the applicability and the characteristic of each analytical method. Conclusively, the aim is to provide the guidance for researchers to utilize the most appropriate analytical tool to determine the KD values." @default.
- W2801253218 created "2018-05-17" @default.
- W2801253218 creator A5020026766 @default.
- W2801253218 creator A5022484632 @default.
- W2801253218 creator A5076799529 @default.
- W2801253218 date "2018-06-01" @default.
- W2801253218 modified "2023-09-25" @default.
- W2801253218 title "Overview of the detection methods for equilibrium dissociation constant KD of drug-receptor interaction" @default.
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