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- W2802116543 endingPage "88" @default.
- W2802116543 startingPage "71" @default.
- W2802116543 abstract "Research on GPR34, which was discovered in 1999 as an orphan G protein-coupled receptor of the rhodopsin-like class, disclosed its physiologic relevance only piece by piece. Being present in all recent vertebrate genomes analyzed so far it seems to improve the fitness of species although it is not essential for life and reproduction as GPR34-deficient mice demonstrate. However, closer inspection of macrophages and microglia, where it is mainly expressed, revealed its relevance in immune cell function. Recent data clearly demonstrate that GPR34 function is required to arrest microglia in the M0 homeostatic non-phagocytic phenotype. Herein, we summarize the current knowledge on its evolution, genomic and structural organization, physiology, pharmacology and relevance in human diseases including neurodegenerative diseases and cancer, which accumulated over the last 20 years." @default.
- W2802116543 created "2018-05-17" @default.
- W2802116543 creator A5002097111 @default.
- W2802116543 creator A5054876758 @default.
- W2802116543 creator A5060811223 @default.
- W2802116543 creator A5063460244 @default.
- W2802116543 date "2018-09-01" @default.
- W2802116543 modified "2023-10-02" @default.
- W2802116543 title "The G protein-coupled receptor GPR34 – The past 20 years of a grownup" @default.
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