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- W2802833423 abstract "We identified novel (3R, 5S)-3-aminomethyl-5-methanesulfanyl hexanoic acid (5a: DS75091588) and (3R, 5S)-3-aminomethyl-5-ethanesulfanyl hexanoic acid (6a: DS18430756) as sulfur-containing γ-amino acid derivatives that were useful for the treatment of neuropathic pain. These two compounds exhibited a potent analgesic effect in animal models of both type I diabetes and type II diabetes, and good pharmacokinetics." @default.
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- W2802833423 date "2018-06-01" @default.
- W2802833423 modified "2023-10-05" @default.
- W2802833423 title "Alkylsulfanyl analogs as potent α 2 δ ligands" @default.
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- W2802833423 doi "https://doi.org/10.1016/j.bmcl.2018.05.006" @default.
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