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- W2803268527 endingPage "1717" @default.
- W2803268527 startingPage "1705" @default.
- W2803268527 abstract "Inhaled administration is underutilised because the drug discovery process is viewed as challenging, risky, and expensive. However, unmet medical need continues to grow, and significant opportunities exist to discover novel inhaled medicines delivering the required lung concentrations while minimising systemic exposure. This profile could be achieved by a combination of properties, including lung retention and low oral bioavailability. Property-based rules exist for orally administered compounds, but there has been limited progress defining in silico predictors to guide the discovery of novel inhaled drugs. Recently, the use of informative cell- and tissue-based screens has greatly facilitated the identification of compounds with optimal characteristics for inhaled delivery. Here, we address opportunities for novel inhaled drugs, and the key challenges and uncertainties hampering progress." @default.
- W2803268527 created "2018-06-01" @default.
- W2803268527 creator A5017985797 @default.
- W2803268527 creator A5040751152 @default.
- W2803268527 creator A5049491293 @default.
- W2803268527 creator A5067448740 @default.
- W2803268527 date "2018-10-01" @default.
- W2803268527 modified "2023-10-02" @default.
- W2803268527 title "Current approaches to the discovery of novel inhaled medicines" @default.
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