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- W2805709488 abstract "[Despite as a major inhibitor of urokinase (uPA), paradoxically,] Plasminogen activator inhibitor-1 (PAI-1) has been validated to be highly expressed in various types of tumor biopsy tissues or plasma compared with controls based on huge clinical data bases analysis, more importantly, PAI-1 alone or in conjunction with uPA have been identified as prognostic for disease progression and relapse in certain cancer types. particularly in breast cancer. In addition to play important roles in cell adhesion, migration and invasion, PAI-1 has been reported to induce tumor vascularization and thus promote cell dissemination and tumor metastasis. Furthermore, there are many tumor promoting factors involved in the modulation of PAI-1 expression and activity, which will strengthen the pro-tumorigenic roles of PAI-1. Undoubtedly, PAI-1 may be a promising target for therapeutic intervention of specific cancer treatment. In fact, some PAI-1 inhibitors are currently being evaluated in cancer therapy, which may be developed to new antitumor agents in the future." @default.
- W2805709488 created "2018-06-13" @default.
- W2805709488 creator A5047305117 @default.
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- W2805709488 creator A5064049313 @default.
- W2805709488 creator A5084133517 @default.
- W2805709488 creator A5087327887 @default.
- W2805709488 date "2018-09-01" @default.
- W2805709488 modified "2023-10-16" @default.
- W2805709488 title "Plasminogen activator inhibitor-1 in cancer research" @default.
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