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- W2806645238 endingPage "1760" @default.
- W2806645238 startingPage "1746" @default.
- W2806645238 abstract "Solute carrier membrane transporters (SLCs) control cell exposure to small-molecule drugs, thereby contributing to drug efficacy and failure and/or adverse effects. Moreover, SLCs are genetically linked to various diseases. Hence, in-depth knowledge of SLC function is fundamental for a better understanding of disease pathophysiology and the drug development process. Given that the model organism Drosophila melanogaster (fruit fly) expresses SLCs, such as for the excretion of endogenous and toxic compounds by the hindgut and Malpighian tubules, equivalent to human intestine and kidney, this system appears to be a promising preclinical model to use to study human SLCs. Here, we systematically compare current knowledge of SLCs in Drosophila and humans and describe the Drosophila model as an innovative tool for drug development." @default.
- W2806645238 created "2018-06-13" @default.
- W2806645238 creator A5040827219 @default.
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- W2806645238 creator A5065181138 @default.
- W2806645238 creator A5066057635 @default.
- W2806645238 creator A5090932782 @default.
- W2806645238 date "2018-10-01" @default.
- W2806645238 modified "2023-09-25" @default.
- W2806645238 title "The fruit fly Drosophila melanogaster as an innovative preclinical ADME model for solute carrier membrane transporters, with consequences for pharmacology and drug therapy" @default.
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