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- W2887016314 endingPage "30" @default.
- W2887016314 startingPage "20" @default.
- W2887016314 abstract "Targeted therapies have changed the landscape of treatments for non-small cell lung cancer (NSCLC). Specific targeted therapies have been approved for NSCLC patients harboring genetic alterations in four oncogenes, and agents targeting additional oncogenic drivers are under investigation. Standard first-line chemotherapy has been supplanted by these targeted therapies due to superior efficacy and lower toxicity. Despite excellent response rates and durable responses in some cases, most patients experience relapse within a few years due to the development of acquired drug resistance. Next generation targeted therapies are being developed to overcome drug resistance and extend the duration of therapy. In this review, we summarize the current treatment strategies for the major targetable oncogenic mutations/alterations in NSCLC and discuss the mechanisms leading to acquired drug resistance." @default.
- W2887016314 created "2018-08-22" @default.
- W2887016314 creator A5037214933 @default.
- W2887016314 creator A5044838791 @default.
- W2887016314 creator A5087906702 @default.
- W2887016314 date "2019-01-01" @default.
- W2887016314 modified "2023-09-23" @default.
- W2887016314 title "Targeting oncogenic drivers in lung cancer: Recent progress, current challenges and future opportunities" @default.
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