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- W2887666565 endingPage "1759" @default.
- W2887666565 startingPage "1745" @default.
- W2887666565 abstract "Protein lysine methyltransferases (PKMTs) are epigenetic regulators that modulate gene transcription and physiological functions by catalyzing the post-translational methylation of specific lysine residues of substrate proteins, such as histones. They are considered to be candidate drugs for the treatment of various diseases, including acute myeloid leukemia, and in the past decade, potent and selective inhibitors of individual PKMTs have been developed. Some are currently under clinical trial. In this review, we will focus on some breakthrough PKMT inhibitors, and discuss chemistry-based methods available for elucidation of the physiological functions of PKMTs and methylated proteins." @default.
- W2887666565 created "2018-08-22" @default.
- W2887666565 creator A5009276668 @default.
- W2887666565 creator A5033725334 @default.
- W2887666565 creator A5066169459 @default.
- W2887666565 date "2018-08-06" @default.
- W2887666565 modified "2023-10-16" @default.
- W2887666565 title "Recent Advances in Chemical Tools for the Regulation and Study of Protein Lysine Methyltransferases" @default.
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