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- W2888183732 abstract "Since their discovery in the early 1950s, macrolide antibiotics have been used in both agriculture and medicine. Specifically, macrolides such as erythromycin and azithromycin have found use as substitutes for β-lactam antibiotics in patients with penicillin allergies. Given the extensive use of this class of antibiotics it is no surprise that resistance has spread among pathogenic bacteria. In these bacteria different mechanisms of resistance have been observed. Frequently observed are alterations in the target of macrolides, i.e. the ribosome, as well as upregulation of efflux pumps. However, drug modification is also increasingly observed. Two classes of enzymes have been implicated in macrolide detoxification: macrolide phosphotransferases and macrolide esterases. In this review, we present a comprehensive overview on what is known about macrolide resistance with an emphasis on the macrolide phosphotransferase and esterase enzymes. Furthermore, we explore how this information can assist in addressing resistance to macrolide antibiotics." @default.
- W2888183732 created "2018-08-31" @default.
- W2888183732 creator A5049136686 @default.
- W2888183732 creator A5055421259 @default.
- W2888183732 creator A5084832728 @default.
- W2888183732 date "2018-08-20" @default.
- W2888183732 modified "2023-10-17" @default.
- W2888183732 title "Look and Outlook on Enzyme-Mediated Macrolide Resistance" @default.
- W2888183732 cites W1162169359 @default.
- W2888183732 cites W1567282410 @default.
- W2888183732 cites W1600598234 @default.
- W2888183732 cites W169459663 @default.
- W2888183732 cites W1748215068 @default.
- W2888183732 cites W1817087658 @default.
- W2888183732 cites W1823117548 @default.
- W2888183732 cites W1844155890 @default.
- W2888183732 cites W1894203925 @default.
- W2888183732 cites W1895007034 @default.
- W2888183732 cites W1903417483 @default.
- W2888183732 cites W1954212025 @default.
- W2888183732 cites W1965342157 @default.
- W2888183732 cites W1966597667 @default.
- W2888183732 cites W1969393758 @default.
- W2888183732 cites W1969655420 @default.
- W2888183732 cites W1970802856 @default.
- W2888183732 cites W1974112253 @default.
- W2888183732 cites W1978039465 @default.
- W2888183732 cites W1980564527 @default.
- W2888183732 cites W1982278009 @default.
- W2888183732 cites W1983534198 @default.
- W2888183732 cites W1986039556 @default.
- W2888183732 cites W1988478675 @default.
- W2888183732 cites W1988907123 @default.
- W2888183732 cites W1994950950 @default.
- W2888183732 cites W1997808887 @default.
- W2888183732 cites W2001703011 @default.
- W2888183732 cites W2002259878 @default.
- W2888183732 cites W2004798786 @default.
- W2888183732 cites W2005791049 @default.
- W2888183732 cites W2011204234 @default.
- W2888183732 cites W2015638139 @default.
- W2888183732 cites W2016595403 @default.
- W2888183732 cites W2018530089 @default.
- W2888183732 cites W2020591349 @default.
- W2888183732 cites W2027053574 @default.
- W2888183732 cites W2027295832 @default.
- W2888183732 cites W2032161209 @default.
- W2888183732 cites W2035321536 @default.
- W2888183732 cites W2039026588 @default.
- W2888183732 cites W2039062180 @default.
- W2888183732 cites W2043158848 @default.
- W2888183732 cites W2045316394 @default.
- W2888183732 cites W2046258407 @default.
- W2888183732 cites W2051558613 @default.
- W2888183732 cites W2053432275 @default.
- W2888183732 cites W2054142295 @default.
- W2888183732 cites W2063919745 @default.
- W2888183732 cites W2065193886 @default.
- W2888183732 cites W2066960769 @default.
- W2888183732 cites W2069684779 @default.
- W2888183732 cites W2076233570 @default.
- W2888183732 cites W2079228339 @default.
- W2888183732 cites W2079916671 @default.
- W2888183732 cites W2080367724 @default.
- W2888183732 cites W2086402273 @default.
- W2888183732 cites W2087630431 @default.
- W2888183732 cites W2090317768 @default.
- W2888183732 cites W2092299098 @default.
- W2888183732 cites W2092913999 @default.
- W2888183732 cites W2095415823 @default.
- W2888183732 cites W2097618796 @default.
- W2888183732 cites W2098278149 @default.
- W2888183732 cites W2104500040 @default.
- W2888183732 cites W2105289202 @default.
- W2888183732 cites W2105838618 @default.
- W2888183732 cites W2110767549 @default.
- W2888183732 cites W2119278807 @default.
- W2888183732 cites W2119966574 @default.
- W2888183732 cites W2122344148 @default.
- W2888183732 cites W2129491200 @default.
- W2888183732 cites W2132254727 @default.
- W2888183732 cites W2132507709 @default.
- W2888183732 cites W2134167455 @default.
- W2888183732 cites W2135493947 @default.
- W2888183732 cites W2136653513 @default.
- W2888183732 cites W2149548739 @default.
- W2888183732 cites W2153839483 @default.
- W2888183732 cites W2158837823 @default.
- W2888183732 cites W2162371815 @default.
- W2888183732 cites W2162626206 @default.
- W2888183732 cites W2166117980 @default.
- W2888183732 cites W2171076011 @default.
- W2888183732 cites W2199203801 @default.
- W2888183732 cites W2288396081 @default.
- W2888183732 cites W2296806616 @default.
- W2888183732 cites W2325819067 @default.
- W2888183732 cites W2335059016 @default.
- W2888183732 cites W2397201307 @default.
- W2888183732 cites W2398757352 @default.
- W2888183732 cites W2470455431 @default.