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- W2891420275 endingPage "33439" @default.
- W2891420275 startingPage "33416" @default.
- W2891420275 abstract "Interleukin-1 receptor-associated kinases (IRAK1, IRAK2, IRAK3 [IRAK-M], and IRAK4) are serine-threonine kinases involved in toll-like receptor and interleukin-1 signaling pathways, through which they regulate innate immunity and inflammation. Evidence exists that IRAKs play key roles in the pathophysiologies of cancers, and metabolic and inflammatory diseases, and that IRAK inhibition has potential therapeutic benefits. Molecules capable of selectively interfering with IRAK function and expression have been reported, paving the way for the clinical evaluation of IRAK inhibition. Herein, we focus on IRAK1, review its structure and physiological roles, and summarize emerging data for IRAK1 inhibitors in preclinical and clinical studies." @default.
- W2891420275 created "2018-09-27" @default.
- W2891420275 creator A5005050727 @default.
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- W2891420275 creator A5045366442 @default.
- W2891420275 creator A5072336042 @default.
- W2891420275 creator A5076074507 @default.
- W2891420275 creator A5090372525 @default.
- W2891420275 date "2018-09-07" @default.
- W2891420275 modified "2023-10-12" @default.
- W2891420275 title "Inhibition of interleukin-1 receptor-associated kinase 1 (IRAK1) as a therapeutic strategy" @default.
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