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- W2891863973 abstract "목ì 본 ì°êµ¬ë ì¸ê°í¼ë¶ì ì¬ëª¨ë¸(human skin equivalent model, HSEM)ì ì¬ì©íì¬ ë©ë¼ë í©ì±ì í´ì ë¡ ìë ¤ì§ PF3758309ì í¼ë¶ ìê·¹ì±ì ë물ëì²´ìíë²ì ì¼íì¼ë¡ íê°íê³ ì íìë¤. ë°©ë² ì¸ì²´í¼ë¶ì ì¬ì²´ë ì½ë¼ê²ì¼ë¡ ì½í ë matrix insert ìì ì¸ê°ìì ë¶ë¦¬í ê°ì§ì¸í¬(human epidermal keratinocyte, HEK)를 ì±ì¥ ë°°ì§ì í¨ê» ë°°ììì¼ ì ìíìë¤. ì ìë ì¸ê°í¼ë¶ ì ì¬ëª¨ë¸ì ì¬ì©íì¬ PF3758309ì í¼ë¶ ìê·¹ì±(irritation)ì ëí´ì íê°íê³ ì, í´ë¹ 물ì§ì HSEMì ê°ì§ íë©´ ìì ì²ë¦¬í í 3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyltetrazolium bromide (MTT)를 íµíì¬ ì¸í¬ìì¡´ì¨ì 측ì íìë¤. ì¸í¬ìì¡´ì¨ì´ 50% ì´íì¼ ê²½ì° ìê·¹ì±ì´ ì¡´ì¬íë©°, 50% ì´ìì¼ ê²½ì° ë¹ìê·¹ì±ì¼ë¡ íë¨í ì ìë¤. ëí, HSEMì ì´ì©íì¬ PF3758309ì í¼ë¶ ë¶ìì±(corrosion) ë° ë©ë¼ë í©ì± ì í´ë¥ì ê²ì¦íìë¤. ê²°ê³¼ ì ìë HSEMì integrityë epidermal differentiation markersì¸ Keratin 5, Keratin 1, Involucrinì ë°íì ë©´ìì¡°ì§ííì¼ìë²ì¼ë¡ ê²ì¦íìë¤. HSEMì PF3758309를 15 min ëì ì²ë¦¬ í, in vitro irritation assay를 ì§íí ê²°ê³¼, PF3758309ì ì²ë¦¬ ëëê° 0.2, 0.5, 1.0 mg ì¼ ë, ì¸í¬ìì¡´ì¨ì ê°ê° 83.6%, 78.8%, 77.8%ë¡ ëíë¬ì¼ë©°, ìì±ëì¡°êµ°ì¸ 5% sodium dodecyl sulfateì ì²ë¦¬ì ì¸í¬ìì¡´ì¨ 2.8%를 ëíë´ìë¤. ëí, in vitro corrosion assay를 ì§íí ê²°ê³¼, PF3758309ì ì²ë¦¬ ëëê° 0.2, 0.5, 1.0 mg ì¼ ë, ì¸í¬ìì¡´ì¨ì ê°ê° 95.3%, 95.0%, 94.2%ë¡ ëíë¬ë¤. ë¿ë§ ìëë¼, Fontana-Masson ì¼ìë²ì íì©íì¬ PF3758309ê° ì²ë¦¬ë HSEMì ë©ë¼ë ìì¤ì ëì¡°êµ° ëë¹ íì íê² ê°ìë¨ì ë³´ìë¤. ê²°ë¡ ë©ë¼ë í©ì± ì í´ì ë¡ ìë ¤ì§ PF3758309ë í¼ë¶ìê·¹ì±ì´ ììì 본 ì¤íì íµí´ ëíë´ìë¤. íµì¬ì©ì´: ì¸ê°í¼ë¶ì ì¬ëª¨ë¸, PF3758309, ìê·¹, í¼ë¶, ë©ë¼ë í©ì± ì í´" @default.
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- W2891863973 date "2018-08-22" @default.
- W2891863973 modified "2023-10-12" @default.
- W2891863973 title "In Vitro Assessment of Irritation Potential of an Anti-Melanogenic Agent, PF3758309, in a Reconstructed Human Epidermis Model" @default.
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- W2891863973 doi "https://doi.org/10.20402/ajbc.2018.0236" @default.
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