Matches in SemOpenAlex for { <https://semopenalex.org/work/W2892283906> ?p ?o ?g. }
- W2892283906 endingPage "2389" @default.
- W2892283906 startingPage "2374" @default.
- W2892283906 abstract "Chemotherapy based on repeated doses of praziquantel remains the most effective control strategy against schistosomiasis, a neglected tropical disease caused by platyhelminths of the genus Schistosoma spp. Its long-term use, however, raises serious concerns about drug resistance against praziquantel. Therefore, it is generally acknowledged that alternative treatment options are urgently needed. This Review summarizes data on relinquished drugs as well as recent advances in the area of antischistosomal compounds from a medicinal chemistry point of view. Furthermore, insights into the structure-activity relationships of each class of compounds are presented including in vitro and in vivo data, if available. Although many compounds have demonstrated good antischistosomal activity in vitro, they offer little promise to replace praziquantel. Nevertheless, the race to develop novel antischistosomal agents is ongoing." @default.
- W2892283906 created "2018-09-27" @default.
- W2892283906 creator A5016865869 @default.
- W2892283906 creator A5038327163 @default.
- W2892283906 creator A5044780249 @default.
- W2892283906 creator A5063243817 @default.
- W2892283906 creator A5076727775 @default.
- W2892283906 date "2018-11-07" @default.
- W2892283906 modified "2023-10-05" @default.
- W2892283906 title "Chemotherapy for Fighting Schistosomiasis: Past, Present and Future" @default.
- W2892283906 cites W1274037484 @default.
- W2892283906 cites W1512472858 @default.
- W2892283906 cites W1513489828 @default.
- W2892283906 cites W1521207198 @default.
- W2892283906 cites W1632352899 @default.
- W2892283906 cites W1654134025 @default.
- W2892283906 cites W1825132503 @default.
- W2892283906 cites W1941508647 @default.
- W2892283906 cites W1964248507 @default.
- W2892283906 cites W1965260090 @default.
- W2892283906 cites W1965927792 @default.
- W2892283906 cites W1968311626 @default.
- W2892283906 cites W1969597927 @default.
- W2892283906 cites W1970406923 @default.
- W2892283906 cites W1971164927 @default.
- W2892283906 cites W1973935887 @default.
- W2892283906 cites W1976330466 @default.
- W2892283906 cites W1976862160 @default.
- W2892283906 cites W1978342290 @default.
- W2892283906 cites W1978511725 @default.
- W2892283906 cites W1980166733 @default.
- W2892283906 cites W1980757462 @default.
- W2892283906 cites W1981906828 @default.
- W2892283906 cites W1982187630 @default.
- W2892283906 cites W1983094623 @default.
- W2892283906 cites W1984075743 @default.
- W2892283906 cites W1985662676 @default.
- W2892283906 cites W1985678753 @default.
- W2892283906 cites W1985716169 @default.
- W2892283906 cites W1985905543 @default.
- W2892283906 cites W1988687410 @default.
- W2892283906 cites W1990470761 @default.
- W2892283906 cites W1990770244 @default.
- W2892283906 cites W1990959786 @default.
- W2892283906 cites W1991474023 @default.
- W2892283906 cites W1991658714 @default.
- W2892283906 cites W1993176720 @default.
- W2892283906 cites W1993347908 @default.
- W2892283906 cites W1994890976 @default.
- W2892283906 cites W1995093410 @default.
- W2892283906 cites W1997430400 @default.
- W2892283906 cites W1997924662 @default.
- W2892283906 cites W1998604274 @default.
- W2892283906 cites W1998943186 @default.
- W2892283906 cites W1999242544 @default.
- W2892283906 cites W2000367696 @default.
- W2892283906 cites W2000388030 @default.
- W2892283906 cites W2001659849 @default.
- W2892283906 cites W2002759367 @default.
- W2892283906 cites W2002830367 @default.
- W2892283906 cites W2004245077 @default.
- W2892283906 cites W2004918705 @default.
- W2892283906 cites W2005767890 @default.
- W2892283906 cites W2005888303 @default.
- W2892283906 cites W2009972285 @default.
- W2892283906 cites W201152868 @default.
- W2892283906 cites W2013711392 @default.
- W2892283906 cites W2013955914 @default.
- W2892283906 cites W2018377353 @default.
- W2892283906 cites W2018849687 @default.
- W2892283906 cites W2019274918 @default.
- W2892283906 cites W2020024165 @default.
- W2892283906 cites W2021415648 @default.
- W2892283906 cites W2022128328 @default.
- W2892283906 cites W2023374722 @default.
- W2892283906 cites W2025057325 @default.
- W2892283906 cites W2031812119 @default.
- W2892283906 cites W2032475967 @default.
- W2892283906 cites W2032566788 @default.
- W2892283906 cites W2034340491 @default.
- W2892283906 cites W2038178479 @default.
- W2892283906 cites W2038227349 @default.
- W2892283906 cites W2038522404 @default.
- W2892283906 cites W2041375888 @default.
- W2892283906 cites W2044172907 @default.
- W2892283906 cites W2045484078 @default.
- W2892283906 cites W2045965339 @default.
- W2892283906 cites W2046323432 @default.
- W2892283906 cites W2049246241 @default.
- W2892283906 cites W2049433339 @default.
- W2892283906 cites W2050384029 @default.
- W2892283906 cites W2050462153 @default.
- W2892283906 cites W2050700386 @default.
- W2892283906 cites W2052819414 @default.
- W2892283906 cites W2054043786 @default.
- W2892283906 cites W2054873814 @default.
- W2892283906 cites W2055515709 @default.
- W2892283906 cites W2057456599 @default.