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- W2902063722 abstract "FLT3 mutations are one of the most common findings in acute myeloid leukemia (AML). FLT3 inhibitors have been in active clinical development. Midostaurin as the first-in-class FLT3 inhibitor has been approved for treatment of patients with FLT3-mutated AML. In this review, we summarized the preclinical and clinical studies on new FLT3 inhibitors, including sorafenib, lestaurtinib, sunitinib, tandutinib, quizartinib, midostaurin, gilteritinib, crenolanib, cabozantinib, Sel24-B489, G-749, AMG 925, TTT-3002, and FF-10101. New generation FLT3 inhibitors and combination therapies may overcome resistance to first-generation agents." @default.
- W2902063722 created "2018-12-11" @default.
- W2902063722 creator A5012861177 @default.
- W2902063722 creator A5060121746 @default.
- W2902063722 creator A5082590593 @default.
- W2902063722 date "2018-12-01" @default.
- W2902063722 modified "2023-10-15" @default.
- W2902063722 title "FLT3 inhibitors in acute myeloid leukemia" @default.
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