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- W2909093302 endingPage "3042" @default.
- W2909093302 startingPage "3029" @default.
- W2909093302 abstract "The ubiquitous Ca2+ /calmodulin-dependent phosphatase calcineurin is a key regulator of pathological cardiac hypertrophy whose therapeutic targeting in heart disease has been elusive due to its role in other essential biological processes. Calcineurin is targeted to diverse intracellular compartments by association with scaffold proteins, including by multivalent A-kinase anchoring proteins (AKAPs) that bind protein kinase A and other important signalling enzymes determining cardiac myocyte function and phenotype. Calcineurin anchoring by AKAPs confers specificity to calcineurin function in the cardiac myocyte. Targeting of calcineurin 'signalosomes' may provide a rationale for inhibiting the phosphatase in disease." @default.
- W2909093302 created "2019-01-25" @default.
- W2909093302 creator A5014637766 @default.
- W2909093302 creator A5029738376 @default.
- W2909093302 creator A5037031481 @default.
- W2909093302 date "2018-12-26" @default.
- W2909093302 modified "2023-10-14" @default.
- W2909093302 title "Calcineurin–AKAP interactions: therapeutic targeting of a pleiotropic enzyme with a little help from its friends" @default.
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