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- W2912174608 endingPage "151" @default.
- W2912174608 startingPage "130" @default.
- W2912174608 abstract "Cathepsins are an important category of enzymes that have attracted great attention for the delivery of drugs to improve the therapeutic outcome of a broad range of nanoscale drug delivery systems. These proteases can be utilized for instance through actuation of polymer-drug conjugates (e.g., triggering the drug release) to bypass limitations of many drug candidates. A substantial amount of work has been witnessed in the design and the evaluation of Cathepsin-sensitive drug delivery systems, especially based on the tetra-peptide sequence (Gly-Phe-Leu-Gly, GFLG) which has been extensively used as a spacer that can be cleaved in the presence of Cathepsin B. This Review Article will give an in-depth overview of the design and the biological evaluation of Cathepsin-sensitive drug delivery systems and their application in different pathologies including cancer before discussing Cathepsin B-cleavable prodrugs under clinical trials." @default.
- W2912174608 created "2019-02-21" @default.
- W2912174608 creator A5001640643 @default.
- W2912174608 creator A5004817332 @default.
- W2912174608 creator A5060168315 @default.
- W2912174608 date "2019-11-01" @default.
- W2912174608 modified "2023-09-30" @default.
- W2912174608 title "Cathepsin-sensitive nanoscale drug delivery systems for cancer therapy and other diseases" @default.
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