Matches in SemOpenAlex for { <https://semopenalex.org/work/W2912657221> ?p ?o ?g. }
- W2912657221 endingPage "741" @default.
- W2912657221 startingPage "723" @default.
- W2912657221 abstract "Proteolysis-targeting chimeras (PROTACs) are an emerging tool for therapeutic intervention by reducing or eliminating disease-causing proteins. PROTACs are bifunctional molecules that consist of a target protein ligand, a linker and an E3 ligase ligand, which mediate the polyubiquitination of the target protein, ultimately leading to the target protein degradation by the ubiquitin–proteasome pathway. We review some of the main PROTACs that have been reported recently and discuss their potential therapeutic benefits over classical enzyme inhibition. Future research is expected to focus on the delivery and bioavailability of PROTACs due to their high molecular weight (700–1000 Da)." @default.
- W2912657221 created "2019-02-21" @default.
- W2912657221 creator A5001909579 @default.
- W2912657221 creator A5035066936 @default.
- W2912657221 date "2019-04-01" @default.
- W2912657221 modified "2023-09-24" @default.
- W2912657221 title "Proteolysis-targeting chimeras for targeting protein for degradation" @default.
- W2912657221 cites W1486112083 @default.
- W2912657221 cites W1488181101 @default.
- W2912657221 cites W1495575342 @default.
- W2912657221 cites W1512690422 @default.
- W2912657221 cites W1527383154 @default.
- W2912657221 cites W1542410645 @default.
- W2912657221 cites W1565539350 @default.
- W2912657221 cites W1611419331 @default.
- W2912657221 cites W1760302596 @default.
- W2912657221 cites W1968143066 @default.
- W2912657221 cites W1982810302 @default.
- W2912657221 cites W1986231077 @default.
- W2912657221 cites W1988013217 @default.
- W2912657221 cites W1988884933 @default.
- W2912657221 cites W1990735654 @default.
- W2912657221 cites W1994344724 @default.
- W2912657221 cites W1995079678 @default.
- W2912657221 cites W2000000541 @default.
- W2912657221 cites W2001582257 @default.
- W2912657221 cites W2002111767 @default.
- W2912657221 cites W2009693397 @default.
- W2912657221 cites W2009886463 @default.
- W2912657221 cites W2009949436 @default.
- W2912657221 cites W2015273986 @default.
- W2912657221 cites W2015345028 @default.
- W2912657221 cites W2025031463 @default.
- W2912657221 cites W2030689174 @default.
- W2912657221 cites W2037420113 @default.
- W2912657221 cites W2042037931 @default.
- W2912657221 cites W2044423100 @default.
- W2912657221 cites W2048964430 @default.
- W2912657221 cites W2050480410 @default.
- W2912657221 cites W2052268618 @default.
- W2912657221 cites W2052787205 @default.
- W2912657221 cites W2054746486 @default.
- W2912657221 cites W2057460011 @default.
- W2912657221 cites W2071909842 @default.
- W2912657221 cites W2073651093 @default.
- W2912657221 cites W2076647485 @default.
- W2912657221 cites W2077141448 @default.
- W2912657221 cites W2080046473 @default.
- W2912657221 cites W2083469632 @default.
- W2912657221 cites W2084372424 @default.
- W2912657221 cites W2084897147 @default.
- W2912657221 cites W2089103836 @default.
- W2912657221 cites W2089707350 @default.
- W2912657221 cites W2090958270 @default.
- W2912657221 cites W2097933346 @default.
- W2912657221 cites W2101948634 @default.
- W2912657221 cites W2103177037 @default.
- W2912657221 cites W2120572492 @default.
- W2912657221 cites W2130968395 @default.
- W2912657221 cites W2131441324 @default.
- W2912657221 cites W2144855932 @default.
- W2912657221 cites W2151683271 @default.
- W2912657221 cites W2165985213 @default.
- W2912657221 cites W2176682109 @default.
- W2912657221 cites W2227431445 @default.
- W2912657221 cites W2237051895 @default.
- W2912657221 cites W2318148969 @default.
- W2912657221 cites W2409568753 @default.
- W2912657221 cites W2518578896 @default.
- W2912657221 cites W2525068643 @default.
- W2912657221 cites W2530302741 @default.
- W2912657221 cites W2553908226 @default.
- W2912657221 cites W2559947248 @default.
- W2912657221 cites W2561008093 @default.
- W2912657221 cites W2566053885 @default.
- W2912657221 cites W2589026097 @default.
- W2912657221 cites W2593430295 @default.
- W2912657221 cites W2596306432 @default.
- W2912657221 cites W2597078857 @default.
- W2912657221 cites W2604040637 @default.
- W2912657221 cites W2621934513 @default.
- W2912657221 cites W2623602792 @default.
- W2912657221 cites W2625751604 @default.
- W2912657221 cites W2704517448 @default.
- W2912657221 cites W2735419424 @default.
- W2912657221 cites W2743800043 @default.
- W2912657221 cites W2761240402 @default.
- W2912657221 cites W2767856718 @default.
- W2912657221 cites W2778368398 @default.
- W2912657221 cites W2782495371 @default.
- W2912657221 cites W2790815306 @default.
- W2912657221 cites W2792069216 @default.
- W2912657221 cites W2792290561 @default.
- W2912657221 cites W2794265154 @default.
- W2912657221 cites W2794623623 @default.
- W2912657221 cites W2805067921 @default.
- W2912657221 cites W2805296794 @default.
- W2912657221 cites W2806694687 @default.