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- W2925181816 endingPage "1098" @default.
- W2925181816 startingPage "1098" @default.
- W2925181816 abstract "Metabotropic glutamate (mGlu) receptors are a family of eight GPCRs that are attractive drug discovery targets to modulate glutamate action and response. Here we review the application of computational methods to the study of this family of receptors. X-ray structures of the extracellular and 7-transmembrane domains have played an important role to enable structure-based modeling approaches, whilst we also discuss the successful application of ligand-based methods. We summarize the literature and highlight the areas where modeling and experiment have delivered important understanding for mGlu receptor drug discovery. Finally, we offer suggestions of future areas of opportunity for computational work." @default.
- W2925181816 created "2019-04-01" @default.
- W2925181816 creator A5022201149 @default.
- W2925181816 creator A5059097965 @default.
- W2925181816 creator A5078699014 @default.
- W2925181816 date "2019-03-20" @default.
- W2925181816 modified "2023-10-16" @default.
- W2925181816 title "Computational Drug Design Applied to the Study of Metabotropic Glutamate Receptors" @default.
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