Matches in SemOpenAlex for { <https://semopenalex.org/work/W2934123297> ?p ?o ?g. }
- W2934123297 endingPage "721" @default.
- W2934123297 startingPage "707" @default.
- W2934123297 abstract "Targeted covalent modification is assuming consolidated importance in drug discovery. In this context, the electrophilic tuning of redox-dependent cell signaling is attracting major interest, as it opens prospect for treating numerous pathologic conditions. Herein, we discuss the rationale and the issues of electrophile-based approaches, focusing on the transcriptional Nrf2-Keap1 pathway as a test case. We also highlight relevant medicinal chemistry strategies researchers have devised to meet the ambitious goal, dwelling on the investigational and therapeutic potential of modulating redox-signaling networks through regulatory cysteine switches." @default.
- W2934123297 created "2019-04-11" @default.
- W2934123297 creator A5006248681 @default.
- W2934123297 creator A5011047821 @default.
- W2934123297 creator A5023513144 @default.
- W2934123297 creator A5071816363 @default.
- W2934123297 date "2019-04-01" @default.
- W2934123297 modified "2023-10-16" @default.
- W2934123297 title "Lights and shadows of electrophile signaling: focus on the Nrf2-Keap1 pathway" @default.
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