Matches in SemOpenAlex for { <https://semopenalex.org/work/W2947497907> ?p ?o ?g. }
- W2947497907 endingPage "768" @default.
- W2947497907 startingPage "755" @default.
- W2947497907 abstract "Introduction: In pharmaceutical design where future drugs are developed by targeting a specific chosen protein, the evaluation of ligand affinity is crucial. For this very purpose are a multitude of diverse methods which are continuously being improved, which, in turn, makes it difficult to choose which techniques to use in practice. Areas covered: In this review, the authors discuss both experimental and computational approaches for affinity evaluation. Basic principles, general limitations and advantages, as well as main areas of application in drug discovery, are overviewed for some of the most popular ligand binding assays. The authors further provide a guide to affinity predictions, collectively covering several techniques that are used in the first stages of rational drug design. Expert opinion: All affinity estimation methods have limitations and advantages that partially overlap and complement one another. Some of the suggested best practices include cross-verification of data using at least two different techniques and careful data interpretation." @default.
- W2947497907 created "2019-06-07" @default.
- W2947497907 creator A5019080699 @default.
- W2947497907 creator A5036811953 @default.
- W2947497907 creator A5069953531 @default.
- W2947497907 creator A5086452069 @default.
- W2947497907 creator A5089298082 @default.
- W2947497907 date "2019-05-31" @default.
- W2947497907 modified "2023-10-03" @default.
- W2947497907 title "Binding affinity in drug design: experimental and computational techniques" @default.
- W2947497907 cites W1531524766 @default.
- W2947497907 cites W1549357029 @default.
- W2947497907 cites W1573009101 @default.
- W2947497907 cites W1625910593 @default.
- W2947497907 cites W1879205842 @default.
- W2947497907 cites W1967348240 @default.
- W2947497907 cites W1968482666 @default.
- W2947497907 cites W1972650408 @default.
- W2947497907 cites W1985034086 @default.
- W2947497907 cites W1987012451 @default.
- W2947497907 cites W1996235332 @default.
- W2947497907 cites W1996634962 @default.
- W2947497907 cites W2009529127 @default.
- W2947497907 cites W2012208164 @default.
- W2947497907 cites W2019466240 @default.
- W2947497907 cites W2022868541 @default.
- W2947497907 cites W2027279463 @default.
- W2947497907 cites W2028035578 @default.
- W2947497907 cites W2032371840 @default.
- W2947497907 cites W2032579758 @default.
- W2947497907 cites W2033757486 @default.
- W2947497907 cites W2034078233 @default.
- W2947497907 cites W2036108598 @default.
- W2947497907 cites W2036140802 @default.
- W2947497907 cites W2043604722 @default.
- W2947497907 cites W2047132220 @default.
- W2947497907 cites W2047730466 @default.
- W2947497907 cites W2054461066 @default.
- W2947497907 cites W2055039476 @default.
- W2947497907 cites W2057806291 @default.
- W2947497907 cites W2063644741 @default.
- W2947497907 cites W2066122522 @default.
- W2947497907 cites W2067778660 @default.
- W2947497907 cites W2071484335 @default.
- W2947497907 cites W2073021822 @default.
- W2947497907 cites W2078363230 @default.
- W2947497907 cites W2079949526 @default.
- W2947497907 cites W2080809427 @default.
- W2947497907 cites W2084303627 @default.
- W2947497907 cites W2085829368 @default.
- W2947497907 cites W2087271871 @default.
- W2947497907 cites W2087661061 @default.
- W2947497907 cites W2091752317 @default.
- W2947497907 cites W2093313511 @default.
- W2947497907 cites W2095719702 @default.
- W2947497907 cites W2107923755 @default.
- W2947497907 cites W2108886196 @default.
- W2947497907 cites W2112154906 @default.
- W2947497907 cites W2117676629 @default.
- W2947497907 cites W2122174098 @default.
- W2947497907 cites W2128332459 @default.
- W2947497907 cites W2134450203 @default.
- W2947497907 cites W2138337932 @default.
- W2947497907 cites W2142820798 @default.
- W2947497907 cites W2142928298 @default.
- W2947497907 cites W2146103350 @default.
- W2947497907 cites W2148950790 @default.
- W2947497907 cites W2149655632 @default.
- W2947497907 cites W2150265183 @default.
- W2947497907 cites W2150862081 @default.
- W2947497907 cites W2151919617 @default.
- W2947497907 cites W2152495850 @default.
- W2947497907 cites W2153207080 @default.
- W2947497907 cites W2154654162 @default.
- W2947497907 cites W2158789571 @default.
- W2947497907 cites W2159367911 @default.
- W2947497907 cites W2171830166 @default.
- W2947497907 cites W2176553778 @default.
- W2947497907 cites W2194538548 @default.
- W2947497907 cites W2275843686 @default.
- W2947497907 cites W2283677448 @default.
- W2947497907 cites W2321635162 @default.
- W2947497907 cites W2335804930 @default.
- W2947497907 cites W2402625670 @default.
- W2947497907 cites W2409721639 @default.
- W2947497907 cites W2470598491 @default.
- W2947497907 cites W2475917031 @default.
- W2947497907 cites W2480097450 @default.
- W2947497907 cites W2508767729 @default.
- W2947497907 cites W2532933839 @default.
- W2947497907 cites W2550887636 @default.
- W2947497907 cites W2557620879 @default.
- W2947497907 cites W2567231876 @default.
- W2947497907 cites W2578119541 @default.
- W2947497907 cites W2582933288 @default.
- W2947497907 cites W2591309385 @default.
- W2947497907 cites W2609589855 @default.
- W2947497907 cites W2625345109 @default.