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- W2950738412 abstract "Abstract Thymic stromal lymphopoietin (TSLP) plays an important role in the differentiation and proliferation of Th2 cells, resulting in eosinophilic inflammation and numerous allergic diseases. Baicalein ( 1 ), a major component of Scutellaria baicalensis , was found to be the first small molecule to block TSLP signaling pathways. It inhibited effectively eosinophil infiltration in house dust mite-induced and ovalbumin-challenged mouse models. Structure-activity relationship studies identified compound 11a , a biphenyl flavanone analog, as a novel human TSLP inhibitor for the discovery and development of new anti-allergic drugs." @default.
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- W2950738412 date "2019-06-19" @default.
- W2950738412 modified "2023-10-12" @default.
- W2950738412 title "Structure-Activity Relationships of Baicalein and its Analogs as Novel TSLP Inhibitors" @default.
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- W2950738412 doi "https://doi.org/10.1038/s41598-019-44853-5" @default.
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