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- W2951716321 abstract "Synthesis and ability to displace [3H]diazepam binding from rat brain membranes of the 3-(alkoxycarbonyl)-4H-pyrimido[2,1-b]benzothiazol-4-ones 3a–p and related compounds 10–12 are described. It has been found that some compounds bind to the benzodiazepine receptor (BZR) with potency greater than chlordiazepoxide. From a structure-affinity point of view the substitution at 6-position of pyrimido [2,1-b]benzothiazole nucleus was found conductive to higher affinity. In vitro data (GABA ratio) lend support to the fact that the most active compounds 3j, 1 might posses agonist properties at BZR." @default.
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- W2951716321 date "1992-01-01" @default.
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- W2951716321 title "Synthesis and benzodiazepine receptor binding of some 4H-pyrimido[2,1-b]benzothiazol-4-ones" @default.
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- W2951716321 doi "https://doi.org/10.1016/0223-5234(92)90058-9" @default.
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