Matches in SemOpenAlex for { <https://semopenalex.org/work/W2956534958> ?p ?o ?g. }
- W2956534958 endingPage "1288" @default.
- W2956534958 startingPage "1276" @default.
- W2956534958 abstract "C-Met, also referred to as Hepatocyte Growth Factor Receptor (HGFR), is a heterodimeric receptor tyrosine kinase. It has been determined that c-Met gene mutations, overexpression, and amplification also occur in a variety of human tumor types, and these events are closely related to the aberrant activation of the HGF/c-Met signaling pathway. Meanwhile, high c-Met expression is closely associated with poor prognosis in cancer patients. The c-Met kinase has emerged as an attractive target for developing antitumor agents. In this review, we cover the recent advances on the small molecule c-Met inhibitors discovered from 2018 until now, with a main focus on the rational design, synthesis and structureactivity relationship analysis." @default.
- W2956534958 created "2019-07-23" @default.
- W2956534958 creator A5061890892 @default.
- W2956534958 creator A5083457739 @default.
- W2956534958 creator A5091667084 @default.
- W2956534958 date "2019-09-03" @default.
- W2956534958 modified "2023-10-14" @default.
- W2956534958 title "Recent Progress in the Development of Small Molecule c-Met Inhibitors" @default.
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