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- W2959893905 endingPage "2874" @default.
- W2959893905 startingPage "2859" @default.
- W2959893905 abstract "Adenosine is a purine nucleoside which is an effective controller of inflammation. The inflammatory effect of adenosine is expressed via its four receptor subtypes viz. A1, A2A, A2B and A3. The various inflammatory conditions including rheumatoid arthritis (RA) are initiated by adenosine receptors of which A2A and A3 play a vital role. RA primarily is an auto-immune disorder which is manifested as chronic inflammation in the synovial lining of joints. In order to develop an effective treatment, the role of cytokines, IL-1, TNF-α and IL-6 is crucial. Besides, the knowledge of PI3K-PKB/Akt and NF-kB signaling pathway is also important to understand the antiinflammatory targets. Methotrexate along with various other molecules like, NSAIDs and DMARDs are presently used as treatment lines for controlling RA. The enhanced knowledge of the preclinical stages and pathogenesis along with recent potent therapeutics raises the hopes that RA can be prevented in the near future." @default.
- W2959893905 created "2019-07-23" @default.
- W2959893905 creator A5004980618 @default.
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- W2959893905 creator A5015596478 @default.
- W2959893905 creator A5061800324 @default.
- W2959893905 creator A5087728639 @default.
- W2959893905 date "2019-10-09" @default.
- W2959893905 modified "2023-09-27" @default.
- W2959893905 title "Perspective and Potential of A2A and A3 Adenosine Receptors as Therapeutic Targets for the Treatment of Rheumatoid Arthritis" @default.
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