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- W2971513585 abstract "An important factor determining the pharmacological response to antitumor drugs is their concentrations in cancer cells, which accounts for the net interaction with their intracellular molecular targets. Accordingly, mechanisms leading to reduced intracellular levels of active agents play a crucial role in cancer chemoresistance. These include impaired drug uptake through solute carrier (SLC) proteins and efficient drug export by ATP-dependent pumps belonging to the ATP-binding cassette (ABC) superfamily of proteins. Since the net movement of drugs in-and-out the cells depends on the overall expression of carrier proteins, defining the so-called transportome, special attention has been devoted to the study of transcriptome regarding these proteins. Nevertheless, genetic variants affecting SLC and ABC genes may markedly affect the bioavailability and, hence, the efficacy of anticancer drugs." @default.
- W2971513585 created "2019-09-12" @default.
- W2971513585 creator A5004449174 @default.
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- W2971513585 creator A5026869228 @default.
- W2971513585 creator A5060425529 @default.
- W2971513585 creator A5061844974 @default.
- W2971513585 date "2019-08-01" @default.
- W2971513585 modified "2023-10-02" @default.
- W2971513585 title "Role of transportome in the pharmacogenomics of hepatocellular carcinoma and hepatobiliary cancer" @default.
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