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- W2977793452 endingPage "240" @default.
- W2977793452 startingPage "203" @default.
- W2977793452 abstract "Transporters play an important role in the absorption, distribution, metabolism, and excretion (ADME) of drugs. In recent years, various in vitro, in situ/ex vivo, and in vivo methods have been established for studying transporter function and drug-transporter interaction. In this chapter, the major types of in vitro models for drug transport studies comprise membrane-based assays, cell-based assays (such as primary cell cultures, immortalized cell lines), and transporter-transfected cell lines with single transporters or multiple transporters. In situ/ex vivo models comprise isolated and perfused organs or tissues. In vivo models comprise transporter gene knockout models, natural mutant animal models, and humanized animal models. This chapter would be focused on the methods for the study of drug transporters in vitro, in situ/ex vivo, and in vivo. The applications, advantages, or limitations of each model and emerging technologies are also mentioned in this chapter." @default.
- W2977793452 created "2019-10-10" @default.
- W2977793452 creator A5037085860 @default.
- W2977793452 date "2019-01-01" @default.
- W2977793452 modified "2023-10-17" @default.
- W2977793452 title "Current Research Method in Transporter Study" @default.
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