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- W2980631738 endingPage "581" @default.
- W2980631738 startingPage "569" @default.
- W2980631738 abstract "Autophagy, defined as a scavenging process of protein aggregates and damaged organelles mediated by lysosomes, plays a significant role in the quality control of macromolecules and organelles. Since protein kinases are integral to the autophagy process, it is critically important to understand the role of kinases in autophagic regulation. At present, intervention of autophagic processes by small-molecule modulators targeting specific kinases has becoming a reasonable and prevalent strategy for treating several varieties of human disease, especially cancer. In this review, we describe the role of some autophagy-related kinase targets and kinase-mediated phosphorylation mechanisms in autophagy regulation. We also summarize the small-molecule kinase inhibitors/activators of these targets, highlighting the opportunities of these new therapeutic agents." @default.
- W2980631738 created "2019-10-25" @default.
- W2980631738 creator A5003547177 @default.
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- W2980631738 creator A5046081003 @default.
- W2980631738 creator A5048655177 @default.
- W2980631738 creator A5080552560 @default.
- W2980631738 creator A5090815103 @default.
- W2980631738 date "2020-04-01" @default.
- W2980631738 modified "2023-10-15" @default.
- W2980631738 title "Targeting autophagy-related protein kinases for potential therapeutic purpose" @default.
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