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- W2989583470 endingPage "286" @default.
- W2989583470 startingPage "257" @default.
- W2989583470 abstract "Alzheimer’s disease (AD) is an enormous healthcare challenge, and 50 million people are currently suffering from it. There are several pathophysiological mechanisms involved, but cholinesterase inhibitors remained the major target from the last 2–3 decades. Among four available therapeutics (donepezil, rivastigmine, galantamine, and memantine), three of them are cholinesterase inhibitors. Herein, we describe the role of acetylcholine sterase (AChE) and related hypothesis in AD along with the pharmacological and chemical aspects of the available cholinesterase inhibitors. This chapter discusses the development of several congeners and hybrids of available cholinesterase inhibitors along with their binding patterns in enzyme active sites." @default.
- W2989583470 created "2019-12-05" @default.
- W2989583470 creator A5028294587 @default.
- W2989583470 creator A5068258830 @default.
- W2989583470 creator A5082615497 @default.
- W2989583470 date "2019-11-27" @default.
- W2989583470 modified "2023-09-27" @default.
- W2989583470 title "Cholinesterase as a Target for Drug Development in Alzheimer’s Disease" @default.
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