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- W2997756073 abstract "Several fragment based approaches have been established to identify fragments with good ligand efficiencies, but fail to provide insights into efficient fragment linkage, making the drug discovery process complicated. Herein, we report the applicaation of a novel drug discovery approach that generates biol. active compds., known as kinetic target guided synthesis (TGS). An 1,4 dipolar cycloaddition reaction between azides and alkynes was successfully employed for MIF templated screening to identify novel inhibitors of migration inhibitory factor inhibitors (MIF)." @default.
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- W2997756073 date "2014-01-01" @default.
- W2997756073 modified "2023-09-23" @default.
- W2997756073 title "Kinetic target guided synthesis for the identification of macrophage migration inhibitory factor inhibitors (MIF)" @default.
- W2997756073 hasPublicationYear "2014" @default.
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