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- W2999574124 abstract "Abstract The treatment of invasive fungal infections remains challenging due to limitations in currently available antifungal therapies including toxicity, interactions, restricted routes of administration, and drug resistance. This review focuses on novel therapies in clinical development, including drugs and a device. These drugs have novel mechanisms of action to overcome resistance, and some offer new formulations providing distinct advantages over current therapies to improve safety profiles and reduce interactions. Among agents that target the cell wall, 2 glucan synthesis inhibitors are discussed (rezafungin and ibrexafungerp), as well as fosmanogepix and nikkomycin Z. Agents that target the cell membrane include 3 fourth-generation azoles, oral encochleated amphotericin B, and aureobasidin A. Among agents with intracellular targets, we will review olorofim, VL-2397, T-2307, AR-12, and MGCD290. In addition, we will describe neurapheresis, a device used as adjunctive therapy for cryptococcosis. With a field full of novel treatments for fungal infections, the future looks promising." @default.
- W2999574124 created "2020-01-23" @default.
- W2999574124 creator A5028882117 @default.
- W2999574124 creator A5033764045 @default.
- W2999574124 creator A5063549349 @default.
- W2999574124 creator A5077898604 @default.
- W2999574124 date "2020-01-12" @default.
- W2999574124 modified "2023-10-10" @default.
- W2999574124 title "Hope on the Horizon: Novel Fungal Treatments in Development" @default.
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