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- W3009475840 endingPage "7985" @default.
- W3009475840 startingPage "7957" @default.
- W3009475840 abstract "The ubiquitin proteasome system (UPS) presents many opportunities for pharmacological intervention. Key players in the UPS are E3 ubiquitin ligases, responsible for conjugation of ubiquitin to specific cognate substrates. Numbering more than 600 members, these ligases represent the most selective way to intervene within this physiologically important system. This Perspective highlights some of the dedicated medicinal chemistry efforts directed at inhibiting the function of specific single-protein and multicomponent RING-type E3 ubiquitin ligases. We present opportunities and challenges associated with targeting this important class of enzymes." @default.
- W3009475840 created "2020-03-13" @default.
- W3009475840 creator A5013337250 @default.
- W3009475840 creator A5034197003 @default.
- W3009475840 creator A5074676231 @default.
- W3009475840 date "2020-03-06" @default.
- W3009475840 modified "2023-09-25" @default.
- W3009475840 title "Medicinal Chemistry of Inhibiting RING-Type E3 Ubiquitin Ligases" @default.
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