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- W3022303714 abstract "Building on the concepts provided in Chapters 3 and 4 Chapter 3 Chapter 4, this chapter focuses on the mechanism of action of enzyme inhibitors and enzyme inactivators and their consequent usefulness as drugs. With extensive use of examples and case histories, several subcategories of reversible inhibition are covered, including competitive inhibition, stabilization of an enzyme conformation, substrate mimicry, transition state mimicry, and slow, tight-binding inhibition. Irreversible enzyme inhibition, including the subcategories of affinity labeling and mechanism-based inactivation, is discussed with the use of multiple examples." @default.
- W3022303714 created "2020-05-13" @default.
- W3022303714 creator A5036064752 @default.
- W3022303714 date "1992-01-01" @default.
- W3022303714 modified "2023-09-23" @default.
- W3022303714 title "Enzyme Inhibition and Inactivation" @default.
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